General Information of the Compound
Compound ID
CP0556153
Compound Name
5-[4-[(4-amino-1-bicyclo[2.2.2]octanyl)methoxy]-3-fluorophenyl]-7-methylpyrrolo[2,1-f][1,2,4]triazin-2-amine
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Formula
C22H26FN5O
Molecular Weight
395.482
Canonical SMILES
Cc1cc(-c2ccc(OCC34CCC(N)(CC3)CC4)c(F)c2)c2cnc(N)nn12
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InChI
InChI=1S/C22H26FN5O/c1-14-10-16(18-12-26-20(24)27-28(14)18)15-2-3-19(17(23)11-15)29-13-21-4-7-22(25,8-5-21)9-6-21/h2-3,10-12H,4-9,13,25H2,1H3,(H2,24,27)
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InChIKey
NOMVDZUKCKOVTL-UHFFFAOYSA-N
Physicochemical Property
logP
3.85652
Rotatable Bonds
4
Heavy Atom Count
29
Polar Areas
91.46
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
29

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL4792072
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02546, Toll-like receptor 8
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000040 THP-1 Homo sapiens (Human)  1
1
IC50 = 40 nM
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