General Information of the Compound
Compound ID
CP0552528
Compound Name
[(1S,2R,3S,5R,6S,16E,18E,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2S)-2-[3-[[(2R)-3-amino-2-[[(4R,7S,10S,13R,16S,19R)-10-[4-(6-aminohexylcarbamoylamino)butyl]-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carbonyl]amino]-3-oxopropyl]disulfanyl]propanoyl-methylamino]propanoate
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Structure
Formula
C90H123ClN16O21S4
Molecular Weight
1928.786
Canonical SMILES
CO[C@@H]1\C=C\C=C(C)\Cc2cc(OC)c(Cl)c(c2)N(C)C(=O)C[C@H](OC(=O)[C@H](C)N(C)C(=O)CCSSC[C@H](NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@H](N)Cc3ccccc3)C(=O)N[C@@H](Cc3ccc(O)cc3)C(=O)N[C@H](Cc3c[nH]c4ccccc34)C(=O)N[C@@H](CCCCNC(=O)NCCCCCCN)C(=O)N[C@@H]([C@@H](C)O)C(=O)N2)C(N)=O)[C@@]2(C)O[C@H]2[C@H](C)[C@@H]2C[C@@]1(O)NC(=O)O2
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InChI
InChI=1S/C90H123ClN16O21S4/c1-50-22-21-28-71(125-9)90(123)45-70(126-88(122)105-90)51(2)77-89(5,128-77)72(44-74(111)107(7)68-41-56(38-50)42-69(124-8)75(68)91)127-86(120)52(3)106(6)73(110)33-37-129-130-47-65(78(94)112)101-84(118)67-49-132-131-48-66(102-79(113)60(93)39-54-23-13-12-14-24-54)83(117)99-63(40-55-29-31-58(109)32-30-55)81(115)100-64(43-57-46-97-61-26-16-15-25-59(57)61)82(116)98-62(80(114)104-76(53(4)108)85(119)103-67)27-17-20-36-96-87(121)95-35-19-11-10-18-34-92/h12-16,21-26,28-32,41-42,46,51-53,60,62-67,70-72,76-77,97,108-109,123H,10-11,17-20,27,33-40,43-45,47-49,92-93H2,1-9H3,(H2,94,112)(H,98,116)(H,99,117)(H,100,115)(H,101,118)(H,102,113)(H,103,119)(H,104,114)(H,105,122)(H2,95,96,121)/b28-21+,50-22+/t51-,52+,53-,60-,62+,63+,64-,65+,66+,67+,70+,71-,72+,76+,77+,89-,90+/m1/s1
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InChIKey
IVUJYKMCAYKZQP-BOLKIBJUSA-N
Physicochemical Property
logP
4.1716
Rotatable Bonds
34
Heavy Atom Count
132
Polar Areas
552.68
Hydrogen Bond Donor Count
17
Hydrogen Bond Acceptor Count
27
Complexity
132

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 155566365
ChEMBL ID
CHEMBL4587303
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01505, Somatostatin receptor type 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
Ki = 3350 nM
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