General Information of the Compound
Compound ID
CP0552143
Compound Name
3-(3-hydroxyphenyl)-5-[[methyl-[[(2S)-pyrrolidin-2-yl]methyl]amino]methyl]-6-[3-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidin-4-one
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Formula
C27H26F3N5O2
Molecular Weight
509.532
Canonical SMILES
CN(C[C@@H]1CCCN1)Cc1c(cnc2ncn(-c3cccc(O)c3)c(=O)c12)-c1cccc(c1)C(F)(F)F
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InChI
InChI=1S/C27H26F3N5O2/c1-34(14-19-7-4-10-31-19)15-23-22(17-5-2-6-18(11-17)27(28,29)30)13-32-25-24(23)26(37)35(16-33-25)20-8-3-9-21(36)12-20/h2-3,5-6,8-9,11-13,16,19,31,36H,4,7,10,14-15H2,1H3/t19-/m0/s1
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InChIKey
PSQIQBRDMNUHKA-IBGZPJMESA-N
Physicochemical Property
logP
4.3559
Rotatable Bonds
6
Heavy Atom Count
37
Polar Areas
83.28
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
37

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL4798657
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01505, Somatostatin receptor type 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS