General Information of the Compound
Compound ID
CP0543834
Compound Name
(R)-2-[(2S,3S)-3-{4-[5-(4-Cyclopropoxy-benzyl)-2-ethyl-2H-pyrazol-3-yl]-piperidin-1-ylmethyl}-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-3,3-dimethyl-butyric acid
    Show/Hide
Structure
Formula
C37H49FN4O3
Molecular Weight
616.822
Canonical SMILES
CCn1nc(Cc2ccc(OC3CC3)cc2)cc1C1CCN(C[C@H]2CN(C[C@@H]2c2cccc(F)c2)[C@@H](C(O)=O)C(C)(C)C)CC1
    Show/Hide
InChI
InChI=1S/C37H49FN4O3/c1-5-42-34(21-30(39-42)19-25-9-11-31(12-10-25)45-32-13-14-32)26-15-17-40(18-16-26)22-28-23-41(35(36(43)44)37(2,3)4)24-33(28)27-7-6-8-29(38)20-27/h6-12,20-21,26,28,32-33,35H,5,13-19,22-24H2,1-4H3,(H,43,44)/t28-,33+,35-/m0/s1
    Show/Hide
InChIKey
BQQDYTWNFPNXMT-IDLKRKCPSA-N
Physicochemical Property
logP
6.5684
Rotatable Bonds
11
Heavy Atom Count
45
Polar Areas
70.83
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
6
Complexity
45

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 516274
ChEMBL ID
CHEMBL366873
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00903, C-C chemokine receptor type 5
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 0.4 nM
   TI
   LI
   LO
   TS