General Information of the Compound
Compound ID
CP0538451
Compound Name
5-[[(6R)-6-methyl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl]oxy]-N-[3-(trifluoromethyl)phenyl]indole-1-carboxamide
    Show/Hide
Structure
Formula
C24H20F3N5O2
Molecular Weight
467.451
Canonical SMILES
C[C@@H]1Cc2c(CN1)ncnc2Oc1ccc2n(ccc2c1)C(=O)Nc1cccc(c1)C(F)(F)F
    Show/Hide
InChI
InChI=1S/C24H20F3N5O2/c1-14-9-19-20(12-28-14)29-13-30-22(19)34-18-5-6-21-15(10-18)7-8-32(21)23(33)31-17-4-2-3-16(11-17)24(25,26)27/h2-8,10-11,13-14,28H,9,12H2,1H3,(H,31,33)/t14-/m1/s1
    Show/Hide
InChIKey
NSHMANQZSCXBCX-CQSZACIVSA-N
Physicochemical Property
logP
5.3568
Rotatable Bonds
3
Heavy Atom Count
34
Polar Areas
81.07
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
34

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 90718764
ChEMBL ID
CHEMBL3746897
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00864, Vascular endothelial growth factor receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
IC50 = 109 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 23 nM