General Information of the Compound
Compound ID
CP0533703
Compound Name
N'-hydroxy-N-[1-(4-propan-2-ylpiperazin-1-yl)isoquinolin-7-yl]octanediamide
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Structure
Formula
C24H35N5O3
Molecular Weight
441.576
Canonical SMILES
CC(C)N1CCN(CC1)c1nccc2ccc(NC(=O)CCCCCCC(=O)NO)cc12
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InChI
InChI=1S/C24H35N5O3/c1-18(2)28-13-15-29(16-14-28)24-21-17-20(10-9-19(21)11-12-25-24)26-22(30)7-5-3-4-6-8-23(31)27-32/h9-12,17-18,32H,3-8,13-16H2,1-2H3,(H,26,30)(H,27,31)
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InChIKey
KUEFYQRLDVPNAG-UHFFFAOYSA-N
Physicochemical Property
logP
3.5497
Rotatable Bonds
10
Heavy Atom Count
32
Polar Areas
97.8
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
6
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 122184855
ChEMBL ID
CHEMBL3601341
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00991, Histone deacetylase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 41.63 nM
   TI
   LI
   LO
   TS
Protein ID: PT00995, Histone deacetylase 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 36 nM
   TI
   LI
   LO
   TS
Protein ID: PT01213, Histone deacetylase 6
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 25 nM
   TI
   LI
   LO
   TS