General Information of the Compound
Compound ID
CP0513478
Compound Name
(8S,11R,13S,14S,17S)-11-(2-ethyl-1,3-benzoxazol-5-yl)-17-hydroxy-13-methyl-17-prop-1-ynyl-1,2,6,7,8,11,12,14,15,16-decahydrocyclopenta[a]phenanthren-3-one
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Structure
Formula
C30H33NO3
Molecular Weight
455.598
Canonical SMILES
CCc1nc2cc(ccc2o1)[C@H]1C[C@@]2(C)[C@@H](CC[C@@]2(O)C#CC)[C@@H]2CCC3=CC(=O)CCC3=C12
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InChI
InChI=1S/C30H33NO3/c1-4-13-30(33)14-12-24-22-9-6-18-15-20(32)8-10-21(18)28(22)23(17-29(24,30)3)19-7-11-26-25(16-19)31-27(5-2)34-26/h7,11,15-16,22-24,33H,5-6,8-10,12,14,17H2,1-3H3/t22-,23+,24-,29-,30-/m0/s1
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InChIKey
PBRBWYQRHGSGKO-QDFBQLGHSA-N
Physicochemical Property
logP
6.0441
Rotatable Bonds
2
Heavy Atom Count
34
Polar Areas
63.33
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
4
Complexity
34

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 57392560
ChEMBL ID
CHEMBL1950695
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00967, Glucocorticoid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549 Homo sapiens (Human)  1
1
IC50 = 13 nM
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Protein ID: PT01172, Progesterone receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000078 T-47D Homo sapiens (Human)  1
1
IC50 = 65 nM
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