General Information of the Compound
Compound ID
CP0513000
Compound Name
(4S)-2'-(3,6-dihydro-2H-pyran-5-yl)-4'-fluoro-7'-(2-fluoropyridin-3-yl)spiro[5H-1,3-oxazole-4,9'-xanthene]-2-amine
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Structure
Formula
C25H19F2N3O3
Molecular Weight
447.441
Canonical SMILES
NC1=N[C@@]2(CO1)c1cc(ccc1Oc1c(F)cc(cc21)C1=CCCOC1)-c1cccnc1F
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InChI
InChI=1S/C25H19F2N3O3/c26-20-11-16(15-3-2-8-31-12-15)10-19-22(20)33-21-6-5-14(17-4-1-7-29-23(17)27)9-18(21)25(19)13-32-24(28)30-25/h1,3-7,9-11H,2,8,12-13H2,(H2,28,30)/t25-/m0/s1
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InChIKey
JJDOGEHWXAGFKG-VWLOTQADSA-N
Physicochemical Property
logP
4.5247
Rotatable Bonds
2
Heavy Atom Count
33
Polar Areas
78.96
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
6
Complexity
33

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 53464942
SID: 126491066
ChEMBL ID
CHEMBL3354717
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01020, Beta-secretase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
IC50 = 3 nM
   TI
   LI
   LO
   TS
Protein ID: PT00897, Potassium voltage-gated channel subfamily H member 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki > 15000 nM
   TI
   LI
   LO
   TS