General Information of the Compound
Compound ID
CP0502832
Compound Name
4-[4-(N-Substituted-thio-carbamoyl)-1-piperazinyl]-6-methoxy-7-alkoxyamino-quinazoline derivative
    Show/Hide
Structure
Formula
C31H38N8O4
Molecular Weight
586.697
Canonical SMILES
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)C(NCc1ccc2OCOc2c1)=NC#N
    Show/Hide
InChI
InChI=1S/C31H38N8O4/c1-40-27-17-24-25(18-29(27)41-15-5-10-37-8-3-2-4-9-37)35-21-36-30(24)38-11-13-39(14-12-38)31(34-20-32)33-19-23-6-7-26-28(16-23)43-22-42-26/h6-7,16-18,21H,2-5,8-15,19,22H2,1H3,(H,33,34)
    Show/Hide
InChIKey
KQGFBLYLLXKIPF-UHFFFAOYSA-N
Physicochemical Property
logP
3.37078
Rotatable Bonds
9
Heavy Atom Count
43
Polar Areas
120.6
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
10
Complexity
43

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 44394849
ChEMBL ID
CHEMBL186850
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00844, Platelet-derived growth factor receptor beta
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000197 MG-63 Homo sapiens (Human)  2
1
IC50 = 320 nM
   TI
   LI
   LO
   TS
2
IC50 = 590 nM
   TI
   LI
   LO
   TS