General Information of the Compound
Compound ID
CP0497758
Compound Name
US10272079, Compound 85
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Structure
Formula
C102H132Cl8N14O22S4
Molecular Weight
2318.146
Canonical SMILES
CN1C[C@@H](c2cccc(c2)S(=O)(=O)NCCOCCOCCNC(=O)CN(CCOCCOCCN(CC(=O)NCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)CC(=O)NCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)CC(=O)NCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)c2cc(Cl)cc(Cl)c2C1
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InChI
InChI=1S/C102H132Cl8N14O22S4/c1-119-59-87(83-51-75(103)55-95(107)91(83)63-119)71-9-5-13-79(47-71)147(129,130)115-21-31-141-41-37-137-27-17-111-99(125)67-123(68-100(126)112-18-28-138-38-42-142-32-22-116-148(131,132)80-14-6-10-72(48-80)88-60-120(2)64-92-84(88)52-76(104)56-96(92)108)25-35-145-45-46-146-36-26-124(69-101(127)113-19-29-139-39-43-143-33-23-117-149(133,134)81-15-7-11-73(49-81)89-61-121(3)65-93-85(89)53-77(105)57-97(93)109)70-102(128)114-20-30-140-40-44-144-34-24-118-150(135,136)82-16-8-12-74(50-82)90-62-122(4)66-94-86(90)54-78(106)58-98(94)110/h5-16,47-58,87-90,115-118H,17-46,59-70H2,1-4H3,(H,111,125)(H,112,126)(H,113,127)(H,114,128)/t87-,88-,89-,90-/m0/s1
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InChIKey
GDJONCXOXPGVKD-AFILQZQZSA-N
Physicochemical Property
logP
9.6716
Rotatable Bonds
65
Heavy Atom Count
150
Polar Areas
412.82
Hydrogen Bond Donor Count
8
Hydrogen Bond Acceptor Count
28
Complexity
150

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118460826
ChEMBL ID
CHEMBL3905218
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03762, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 794.33 nM
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Protein ID: PT04309, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 1584.89 nM
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   TS