General Information of the Compound
Compound ID
CP0493785
Compound Name
3-(8-((2-chloro-4-methylphenyl)(2-chlorophenyl)methyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-3-yl)pyrrolidin-2-one
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Structure
Formula
C25H28Cl2N2O2
Molecular Weight
459.417
Canonical SMILES
Cc1ccc(C(N2C3CCC2CC(O)(C3)C2CCNC2=O)c2ccccc2Cl)c(Cl)c1
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InChI
InChI=1S/C25H28Cl2N2O2/c1-15-6-9-19(22(27)12-15)23(18-4-2-3-5-21(18)26)29-16-7-8-17(29)14-25(31,13-16)20-10-11-28-24(20)30/h2-6,9,12,16-17,20,23,31H,7-8,10-11,13-14H2,1H3,(H,28,30)
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InChIKey
ZVWINNTVUYULMY-UHFFFAOYSA-N
Physicochemical Property
logP
4.88522
Rotatable Bonds
4
Heavy Atom Count
31
Polar Areas
52.57
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
3
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44574629
ChEMBL ID
CHEMBL506634
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 781 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 3.6 nM
   TI
   LI
   LO
   TS