General Information of the Compound
Compound ID
CP0492247
Compound Name
(R)-2-[(2S,3S)-3-{4-[5-(4-Cyclopropoxy-benzyl)-2-ethyl-2H-pyrazol-3-yl]-piperidin-1-ylmethyl}-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-3-methyl-butyric acid
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Structure
Formula
C36H47FN4O3
Molecular Weight
602.795
Canonical SMILES
CCn1nc(Cc2ccc(OC3CC3)cc2)cc1C1CCN(C[C@H]2CN(C[C@@H]2c2cccc(F)c2)[C@H](C(C)C)C(O)=O)CC1
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InChI
InChI=1S/C36H47FN4O3/c1-4-41-34(20-30(38-41)18-25-8-10-31(11-9-25)44-32-12-13-32)26-14-16-39(17-15-26)21-28-22-40(35(24(2)3)36(42)43)23-33(28)27-6-5-7-29(37)19-27/h5-11,19-20,24,26,28,32-33,35H,4,12-18,21-23H2,1-3H3,(H,42,43)/t28-,33+,35+/m0/s1
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InChIKey
JLVJXUOOJFCQIH-GCFSYYHISA-N
Physicochemical Property
logP
6.1783
Rotatable Bonds
12
Heavy Atom Count
44
Polar Areas
70.83
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
6
Complexity
44

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 516193
ChEMBL ID
CHEMBL176337
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00903, C-C chemokine receptor type 5
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 1 nM
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