General Information of the Compound
Compound ID
CP0488277
Compound Name
N-[5-[(5-chloro-4-pyrazolo[1,5-a]pyridin-3-ylpyrimidin-2-yl)amino]-4-methoxy-2-[4-[2-(methylamino)acetyl]piperazin-1-yl]phenyl]prop-2-enamide
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Structure
Formula
C28H30ClN9O3
Molecular Weight
576.061
Canonical SMILES
CNCC(=O)N1CCN(CC1)c1cc(OC)c(Nc2ncc(Cl)c(n2)-c2cnn3ccccc23)cc1NC(=O)C=C
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InChI
InChI=1S/C28H30ClN9O3/c1-4-25(39)33-20-13-21(24(41-3)14-23(20)36-9-11-37(12-10-36)26(40)17-30-2)34-28-31-16-19(29)27(35-28)18-15-32-38-8-6-5-7-22(18)38/h4-8,13-16,30H,1,9-12,17H2,2-3H3,(H,33,39)(H,31,34,35)
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InChIKey
SIKCGJIZDJHPPU-UHFFFAOYSA-N
Physicochemical Property
logP
3.1894
Rotatable Bonds
9
Heavy Atom Count
41
Polar Areas
129.02
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
10
Complexity
41

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118719577
ChEMBL ID
CHEMBL3353399
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00922, Epidermal growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000157 NCI-H1975 Homo sapiens (Human)  1
1
IC50 = 66000 nM
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