General Information of the Compound
Compound ID
CP0488090
Compound Name
(E)-4-(dimethylamino)-N-[3-[4-(1H-indazol-3-ylamino)-6-(4-methylpiperazin-1-yl)pyrimidin-2-yl]oxyphenyl]but-2-enamide
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Structure
Formula
C28H33N9O2
Molecular Weight
527.633
Canonical SMILES
CN(C)C\C=C\C(=O)Nc1cccc(Oc2nc(Nc3n[nH]c4ccccc34)cc(n2)N2CCN(C)CC2)c1
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InChI
InChI=1S/C28H33N9O2/c1-35(2)13-7-12-26(38)29-20-8-6-9-21(18-20)39-28-31-24(19-25(32-28)37-16-14-36(3)15-17-37)30-27-22-10-4-5-11-23(22)33-34-27/h4-12,18-19H,13-17H2,1-3H3,(H,29,38)(H2,30,31,32,33,34)/b12-7+
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InChIKey
ADAREYJDNCHIMX-KPKJPENVSA-N
Physicochemical Property
logP
3.6969
Rotatable Bonds
9
Heavy Atom Count
39
Polar Areas
114.54
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
9
Complexity
39

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 122186152
ChEMBL ID
CHEMBL3604939
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00922, Epidermal growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  3
1
IC50 = 700 nM
   TI
   LI
   LO
   TS
2
IC50 = 3600 nM
   TI
   LI
   LO
   TS
3
IC50 = 6700 nM
   TI
   LI
   LO
   TS