General Information of the Compound
Compound ID
CP0482428
Compound Name
N-[1-[1-[(3,5-difluorophenyl)methyl]imidazol-2-yl]-2-(7-methyl-1H-indazol-5-yl)ethyl]-4-(2-oxo-1,4-dihydroquinazolin-3-yl)piperidine-1-carboxamide
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Structure
Formula
C34H34F2N8O2
Molecular Weight
624.696
Canonical SMILES
Cc1cc(CC(NC(=O)N2CCC(CC2)N2Cc3ccccc3NC2=O)c2nccn2Cc2cc(F)cc(F)c2)cc2cn[nH]c12
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InChI
InChI=1S/C34H34F2N8O2/c1-21-12-22(13-25-18-38-41-31(21)25)16-30(32-37-8-11-43(32)19-23-14-26(35)17-27(36)15-23)40-33(45)42-9-6-28(7-10-42)44-20-24-4-2-3-5-29(24)39-34(44)46/h2-5,8,11-15,17-18,28,30H,6-7,9-10,16,19-20H2,1H3,(H,38,41)(H,39,46)(H,40,45)
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InChIKey
IKZZTJAJWRXLNM-UHFFFAOYSA-N
Physicochemical Property
logP
5.89982
Rotatable Bonds
7
Heavy Atom Count
46
Polar Areas
111.18
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
5
Complexity
46

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 11411030
SID: 16506699
ChEMBL ID
CHEMBL2430178
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01670, Calcitonin gene-related peptide type 1 receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000074 SK-N-MC Homo sapiens (Human)  1
1
IC50 = 0.39 nM
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