General Information of the Compound
Compound ID
CP0467848
Compound Name
US10272079, Compound 172
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Structure
Formula
C80H105Cl6N13O19S3
Molecular Weight
1861.711
Canonical SMILES
CN1C[C@@H](c2cccc(c2)S(=O)(=O)NCCOCCOCCNC(=O)NCCC(CCNC(=O)NCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)(CCNC(=O)NCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)NC(=O)COCC(O)=O)c2cc(Cl)cc(Cl)c2C1
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InChI
InChI=1S/C80H105Cl6N13O19S3/c1-97-46-66(63-40-57(81)43-72(84)69(63)49-97)54-7-4-10-60(37-54)119(106,107)93-22-28-115-34-31-112-25-19-90-77(103)87-16-13-80(96-75(100)52-118-53-76(101)102,14-17-88-78(104)91-20-26-113-32-35-116-29-23-94-120(108,109)61-11-5-8-55(38-61)67-47-98(2)50-70-64(67)41-58(82)44-73(70)85)15-18-89-79(105)92-21-27-114-33-36-117-30-24-95-121(110,111)62-12-6-9-56(39-62)68-48-99(3)51-71-65(68)42-59(83)45-74(71)86/h4-12,37-45,66-68,93-95H,13-36,46-53H2,1-3H3,(H,96,100)(H,101,102)(H2,87,90,103)(H2,88,91,104)(H2,89,92,105)/t66-,67-,68-/m0/s1
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InChIKey
IRGWXUXANDOFHM-NLXGDKCYSA-N
Physicochemical Property
logP
7.6979
Rotatable Bonds
50
Heavy Atom Count
121
Polar Areas
402.63
Hydrogen Bond Donor Count
11
Hydrogen Bond Acceptor Count
21
Complexity
121

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 86272299
ChEMBL ID
CHEMBL3983258
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT04309, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 6.31 nM
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Protein ID: PT03762, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 79.43 nM
   TI
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   TS