General Information of the Compound
Compound ID
CP0467846
Compound Name
US10272079, Compound 148
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Structure
Formula
C50H64Cl4N6O12S2
Molecular Weight
1147.038
Canonical SMILES
CN(C)[C@H]1Cc2c(cc(Cl)cc2Cl)[C@@H]1Oc1ccc(cc1)S(=O)(=O)NCCOCCOCCNC(=O)CCC(=O)NCCOCCOCCNS(=O)(=O)c1ccc(O[C@@H]2[C@H](Cc3c2cc(Cl)cc3Cl)N(C)C)cc1
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InChI
InChI=1S/C50H64Cl4N6O12S2/c1-59(2)45-31-39-41(27-33(51)29-43(39)53)49(45)71-35-5-9-37(10-6-35)73(63,64)57-17-21-69-25-23-67-19-15-55-47(61)13-14-48(62)56-16-20-68-24-26-70-22-18-58-74(65,66)38-11-7-36(8-12-38)72-50-42-28-34(52)30-44(54)40(42)32-46(50)60(3)4/h5-12,27-30,45-46,49-50,57-58H,13-26,31-32H2,1-4H3,(H,55,61)(H,56,62)/t45-,46-,49-,50-/m0/s1
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InChIKey
BJMZTIXUXWQYIF-UZYAJYSRSA-N
Physicochemical Property
logP
5.8488
Rotatable Bonds
31
Heavy Atom Count
74
Polar Areas
212.4
Hydrogen Bond Donor Count
4
Hydrogen Bond Acceptor Count
14
Complexity
74

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 90077898
ChEMBL ID
CHEMBL3940439
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT04309, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 3.981 nM
   TI
   LI
   LO
   TS
Protein ID: PT03762, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 15.85 nM
   TI
   LI
   LO
   TS