General Information of the Compound
Compound ID
CP0459555
Compound Name
3-[[7-[2-(dimethylamino)ethoxy]-6-methoxyquinazolin-4-yl]amino]-4-fluoro-2-methylphenol
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Structure
Formula
C20H23FN4O3
Molecular Weight
386.427
Canonical SMILES
COc1cc2c(Nc3c(F)ccc(O)c3C)ncnc2cc1OCCN(C)C
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InChI
InChI=1S/C20H23FN4O3/c1-12-16(26)6-5-14(21)19(12)24-20-13-9-17(27-4)18(28-8-7-25(2)3)10-15(13)22-11-23-20/h5-6,9-11,26H,7-8H2,1-4H3,(H,22,23,24)
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InChIKey
OMKGWBMUCLVMLL-UHFFFAOYSA-N
Physicochemical Property
logP
3.47552
Rotatable Bonds
7
Heavy Atom Count
28
Polar Areas
79.74
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
28

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118112037
ChEMBL ID
CHEMBL3799264
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00864, Vascular endothelial growth factor receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
IC50 > 10000 nM
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