General Information of the Compound
Compound ID
CP0458529
Compound Name
5,8-dichloro-7-(3,5-dimethyl-1,2-oxazol-4-yl)-2-[(4-methoxy-6-methyl-2-oxo-1H-pyridin-3-yl)methyl]-3,4-dihydroisoquinolin-1-one
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Synonyms
PMID28394193-Compound-47
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Structure
Formula
C22H21Cl2N3O4
Molecular Weight
462.333
Canonical SMILES
COc1cc(C)[nH]c(=O)c1CN1CCc2c(Cl)cc(-c3c(C)noc3C)c(Cl)c2C1=O
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InChI
InChI=1S/C22H21Cl2N3O4/c1-10-7-17(30-4)15(21(28)25-10)9-27-6-5-13-16(23)8-14(20(24)19(13)22(27)29)18-11(2)26-31-12(18)3/h7-8H,5-6,9H2,1-4H3,(H,25,28)
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InChIKey
HCXPMZKLLCLZQX-UHFFFAOYSA-N
Physicochemical Property
logP
4.46906
Rotatable Bonds
4
Heavy Atom Count
31
Polar Areas
88.43
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
5
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118616529
ChEMBL ID
CHEMBL4082565
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03003, Histone-lysine N-methyltransferase EZH2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000180 Karpas-422 Homo sapiens (Human)  1
1
IC50 = 8 nM
   TI
   LI
   LO
   TS
Clinical Information about the Compound
Drug 1 ( PMID28394193-Compound-47 )
Drug Name PMID28394193-Compound-47
Company PFIZER INC
Target(s)
Enhancer of zeste homolog 2 (EZH2)
Inhibitor