General Information of the Compound
Compound ID
CP0454462
Compound Name
(2R,3R,4S,5R)-2-[2-chloro-6-[[(3R)-oxolan-3-yl]amino]purin-9-yl]-5-[(3,5-dimethylpyrazol-1-yl)methyl]oxolane-3,4-diol
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Structure
Formula
C19H24ClN7O4
Molecular Weight
449.899
Canonical SMILES
Cc1cc(C)n(C[C@H]2O[C@H]([C@H](O)[C@@H]2O)n2cnc3c(N[C@@H]4CCOC4)nc(Cl)nc23)n1
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InChI
InChI=1S/C19H24ClN7O4/c1-9-5-10(2)27(25-9)6-12-14(28)15(29)18(31-12)26-8-21-13-16(22-11-3-4-30-7-11)23-19(20)24-17(13)26/h5,8,11-12,14-15,18,28-29H,3-4,6-7H2,1-2H3,(H,22,23,24)/t11-,12-,14-,15-,18-/m1/s1
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InChIKey
RBFWIGCXCSBGDT-AJKMGBEJSA-N
Physicochemical Property
logP
0.81324
Rotatable Bonds
5
Heavy Atom Count
31
Polar Areas
132.37
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
11
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 137632488
ChEMBL ID
CHEMBL4067452
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00840, Adenosine receptor A1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 438 nM
   TI
   LI
   LO
   TS
Protein ID: PT00862, Adenosine receptor A2a
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 11900 nM
   TI
   LI
   LO
   TS
Protein ID: PT01278, Adenosine receptor A2b
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 > 60000 nM
   TI
   LI
   LO
   TS
Protein ID: PT01279, Adenosine receptor A3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 996 nM
   TI
   LI
   LO
   TS