General Information of the Compound
Compound ID
CP0453423
Compound Name
4-{7-[2-(1,1-Dioxo-1lambda*6*-thiomorpholin-4-yl)-ethoxy]-6-methoxy-quinazolin-4-yl}-piperazine-1-carboxylic acid (4-isopropoxy-phenyl)-amide
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Structure
Formula
C29H38N6O6S
Molecular Weight
598.726
Canonical SMILES
COc1cc2c(ncnc2cc1OCCN1CCS(=O)(=O)CC1)N1CCN(CC1)C(=O)Nc1ccc(OC(C)C)cc1
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InChI
InChI=1S/C29H38N6O6S/c1-21(2)41-23-6-4-22(5-7-23)32-29(36)35-10-8-34(9-11-35)28-24-18-26(39-3)27(19-25(24)30-20-31-28)40-15-12-33-13-16-42(37,38)17-14-33/h4-7,18-21H,8-17H2,1-3H3,(H,32,36)
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InChIKey
OYRLHMGUQQVGPI-UHFFFAOYSA-N
Physicochemical Property
logP
2.8889
Rotatable Bonds
9
Heavy Atom Count
42
Polar Areas
126.43
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
10
Complexity
42

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 11006502
SID: 16066829
ChEMBL ID
CHEMBL124313
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00844, Platelet-derived growth factor receptor beta
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000197 MG-63 Homo sapiens (Human)  2
1
IC50 = 494 nM
   TI
   LI
   LO
   TS
2
IC50 = 680 nM
   TI
   LI
   LO
   TS