General Information of the Compound
Compound ID
CP0453322
Compound Name
4-{6-Methoxy-7-[3-(3-methyl-butane-1-sulfonyl)-propoxy]-quinazolin-4-yl}-piperazine-1-carboxylic acid (4-isopropoxy-phenyl)-amide
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Structure
Formula
C31H43N5O6S
Molecular Weight
613.781
Canonical SMILES
COc1cc2c(ncnc2cc1OCCCS(=O)(=O)CCC(C)C)N1CCN(CC1)C(=O)Nc1ccc(OC(C)C)cc1
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InChI
InChI=1S/C31H43N5O6S/c1-22(2)11-18-43(38,39)17-6-16-41-29-20-27-26(19-28(29)40-5)30(33-21-32-27)35-12-14-36(15-13-35)31(37)34-24-7-9-25(10-8-24)42-23(3)4/h7-10,19-23H,6,11-18H2,1-5H3,(H,34,37)
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InChIKey
WTFQTDJXZDGOHR-UHFFFAOYSA-N
Physicochemical Property
logP
5.0095
Rotatable Bonds
13
Heavy Atom Count
43
Polar Areas
123.19
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
9
Complexity
43

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44349292
ChEMBL ID
CHEMBL339403
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00844, Platelet-derived growth factor receptor beta
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000197 MG-63 Homo sapiens (Human)  2
1
IC50 = 50 nM
   TI
   LI
   LO
   TS
2
IC50 = 240 nM
   TI
   LI
   LO
   TS