General Information of the Compound
Compound ID
CP0451841
Compound Name
4-[4-(N-Substituted-thio-carbamoyl)-1-piperazinyl]-6-methoxy-7-alkoxyamino-quinazoline derivative
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Structure
Formula
C28H37N9O3
Molecular Weight
547.664
Canonical SMILES
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)C(NCc1cc(C)on1)=NC#N
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InChI
InChI=1S/C28H37N9O3/c1-21-15-22(34-40-21)18-30-28(31-19-29)37-12-10-36(11-13-37)27-23-16-25(38-2)26(17-24(23)32-20-33-27)39-14-6-9-35-7-4-3-5-8-35/h15-17,20H,3-14,18H2,1-2H3,(H,30,31)
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InChIKey
SQQXZLDWWFORTO-UHFFFAOYSA-N
Physicochemical Property
logP
2.9385
Rotatable Bonds
9
Heavy Atom Count
40
Polar Areas
128.17
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
10
Complexity
40

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44394853
ChEMBL ID
CHEMBL186698
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00844, Platelet-derived growth factor receptor beta
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000197 MG-63 Homo sapiens (Human)  2
1
IC50 = 2370 nM
   TI
   LI
   LO
   TS
2
IC50 = 10450 nM
   TI
   LI
   LO
   TS