General Information of the Compound
Compound ID
CP0451088
Compound Name
N-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-4-methyl-3-[(4-thiophen-2-ylpyrimidin-2-yl)amino]benzamide
    Show/Hide
Formula
C29H31N5O3S
Molecular Weight
529.666
Canonical SMILES
COc1cc2CCN(CCNC(=O)c3ccc(C)c(Nc4nccc(n4)-c4cccs4)c3)Cc2cc1OC
    Show/Hide
InChI
InChI=1S/C29H31N5O3S/c1-19-6-7-21(15-24(19)33-29-31-10-8-23(32-29)27-5-4-14-38-27)28(35)30-11-13-34-12-9-20-16-25(36-2)26(37-3)17-22(20)18-34/h4-8,10,14-17H,9,11-13,18H2,1-3H3,(H,30,35)(H,31,32,33)
    Show/Hide
InChIKey
ZBHYVGXHFABTBU-UHFFFAOYSA-N
Physicochemical Property
logP
5.06242
Rotatable Bonds
9
Heavy Atom Count
38
Polar Areas
88.61
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
8
Complexity
38

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
ChEMBL ID
CHEMBL4873838
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01546, ATP-dependent translocase ABCB1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000137 K562/A02 Homo sapiens (Human)  1
1
IC50 = 940 nM
   TI
   LI
   LO
   TS