General Information of the Compound
Compound ID
CP0445631
Compound Name
[(19S)-10,19-diethyl-7-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl] 12-(hydroxyamino)-12-oxododecanoate
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Structure
Formula
C34H41N3O8
Molecular Weight
619.715
Canonical SMILES
CCc1c2Cn3c(cc4c(COC(=O)[C@@]4(CC)OC(=O)CCCCCCCCCCC(=O)NO)c3=O)-c2nc2ccc(O)cc12
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InChI
InChI=1S/C34H41N3O8/c1-3-22-23-17-21(38)15-16-27(23)35-31-24(22)19-37-28(31)18-26-25(32(37)41)20-44-33(42)34(26,4-2)45-30(40)14-12-10-8-6-5-7-9-11-13-29(39)36-43/h15-18,38,43H,3-14,19-20H2,1-2H3,(H,36,39)/t34-/m0/s1
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InChIKey
SLAZSKUYTGFSHH-UMSFTDKQSA-N
Physicochemical Property
logP
5.3049
Rotatable Bonds
14
Heavy Atom Count
45
Polar Areas
157.05
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
10
Complexity
45

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 145982514
ChEMBL ID
CHEMBL4238303
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00991, Histone deacetylase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 12620 nM
   TI
   LI
   LO
   TS
Protein ID: PT00995, Histone deacetylase 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 11780 nM
   TI
   LI
   LO
   TS
Protein ID: PT01213, Histone deacetylase 6
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 1070 nM
   TI
   LI
   LO
   TS