General Information of the Compound
Compound ID
CP0444490
Compound Name
7-(2-amino-3,5-dichloro-6-fluorophenyl)-6-chloro-1-[4,6-di(propan-2-yl)pyrimidin-5-yl]-2-oxo-4-(4-prop-2-enoylpiperazin-1-yl)-1,8-naphthyridine-3-carbonitrile
    Show/Hide
Formula
C32H30Cl3FN8O2
Molecular Weight
684.003
Canonical SMILES
CC(C)c1ncnc(C(C)C)c1-n1c2nc(c(Cl)cc2c(N2CCN(CC2)C(=O)C=C)c(C#N)c1=O)-c1c(N)c(Cl)cc(Cl)c1F
    Show/Hide
InChI
InChI=1S/C32H30Cl3FN8O2/c1-6-22(45)42-7-9-43(10-8-42)29-17-11-21(35)28(23-24(36)19(33)12-20(34)25(23)38)41-31(17)44(32(46)18(29)13-37)30-26(15(2)3)39-14-40-27(30)16(4)5/h6,11-12,14-16H,1,7-10,38H2,2-5H3
    Show/Hide
InChIKey
PXVMFIYXYKYNCY-UHFFFAOYSA-N
Physicochemical Property
logP
6.47728
Rotatable Bonds
6
Heavy Atom Count
46
Polar Areas
134.03
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
9
Complexity
46

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
ChEMBL ID
CHEMBL4857822
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03462, GTPase KRas
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000268 NCI-H358 Homo sapiens (Human)  1
1
IC50 = 18.51 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 4.737 nM