General Information of the Compound
Compound ID
CP0444308
Compound Name
2-[6-[(3R,4S)-3-amino-4-(2,5-difluorophenyl)pyrrolidin-1-yl]pyridin-3-yl]-6-butoxy-3,4-dihydroisoquinolin-1-one
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Structure
Formula
C28H30F2N4O2
Molecular Weight
492.57
Canonical SMILES
CCCCOc1ccc2C(=O)N(CCc2c1)c1ccc(nc1)N1C[C@H](N)[C@H](C1)c1cc(F)ccc1F
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InChI
InChI=1S/C28H30F2N4O2/c1-2-3-12-36-21-6-7-22-18(13-21)10-11-34(28(22)35)20-5-9-27(32-15-20)33-16-24(26(31)17-33)23-14-19(29)4-8-25(23)30/h4-9,13-15,24,26H,2-3,10-12,16-17,31H2,1H3/t24-,26+/m1/s1
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InChIKey
ZMWYWQVZULSCIY-RSXGOPAZSA-N
Physicochemical Property
logP
4.6727
Rotatable Bonds
7
Heavy Atom Count
36
Polar Areas
71.69
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
5
Complexity
36

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 70687361
ChEMBL ID
CHEMBL2011532
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01027, Melanin-concentrating hormone receptor 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 4000 nM
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