General Information of the Compound
Compound ID
CP0444143
Compound Name
US10272079, Compound 74
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Structure
Formula
C72H90Cl6N10O15S3
Molecular Weight
1644.486
Canonical SMILES
CN1C[C@@H](c2cccc(c2)S(=O)(=O)NCCOCCOCCNC(=O)CN(CC(=O)NCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)CC(=O)NCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)c2cc(Cl)cc(Cl)c2C1
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InChI
InChI=1S/C72H90Cl6N10O15S3/c1-85-40-61(58-34-52(73)37-67(76)64(58)43-85)49-7-4-10-55(31-49)104(92,93)82-16-22-101-28-25-98-19-13-79-70(89)46-88(47-71(90)80-14-20-99-26-29-102-23-17-83-105(94,95)56-11-5-8-50(32-56)62-41-86(2)44-65-59(62)35-53(74)38-68(65)77)48-72(91)81-15-21-100-27-30-103-24-18-84-106(96,97)57-12-6-9-51(33-57)63-42-87(3)45-66-60(63)36-54(75)39-69(66)78/h4-12,31-39,61-63,82-84H,13-30,40-48H2,1-3H3,(H,79,89)(H,80,90)(H,81,91)/t61-,62-,63-/m0/s1
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InChIKey
IGEDAVXYMWPIJE-QPUNLCADSA-N
Physicochemical Property
logP
7.3244
Rotatable Bonds
42
Heavy Atom Count
106
Polar Areas
294.15
Hydrogen Bond Donor Count
6
Hydrogen Bond Acceptor Count
19
Complexity
106

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118933974
ChEMBL ID
CHEMBL3920001
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03762, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 158.49 nM
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   TS
Protein ID: PT04309, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS