General Information of the Compound
Compound ID
CP0439514
Compound Name
(8S,11R,13S,14R,17S)-11-(4-dimethylamino-phenyl)-17-(3-dimethylamino-prop-1-ynyl)-17-hydroxy-13-methyl-1,2,8,11,12,13,14,15,16,17-decahydro-6H-7-oxa-cyclopenta[a]phenanthren-3-one
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Structure
Formula
C30H38N2O3
Molecular Weight
474.645
Canonical SMILES
CN(C)CC#C[C@]1(O)CC[C@H]2[C@@H]3OCC4=CC(=O)CCC4=C3[C@H](C[C@]12C)c1ccc(cc1)N(C)C
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InChI
InChI=1S/C30H38N2O3/c1-29-18-25(20-7-9-22(10-8-20)32(4)5)27-24-12-11-23(33)17-21(24)19-35-28(27)26(29)13-15-30(29,34)14-6-16-31(2)3/h7-10,17,25-26,28,34H,11-13,15-16,18-19H2,1-5H3/t25-,26+,28+,29+,30+/m1/s1
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InChIKey
ZOJNIVLVFGPWTA-LXEMEFDRSA-N
Physicochemical Property
logP
3.937
Rotatable Bonds
3
Heavy Atom Count
35
Polar Areas
53.01
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
5
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44425542
ChEMBL ID
CHEMBL231515
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00967, Glucocorticoid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549 Homo sapiens (Human)  1
1
IC50 > 3000 nM
   TI
   LI
   LO
   TS
Protein ID: PT01172, Progesterone receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000078 T-47D Homo sapiens (Human)  1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS