General Information of the Compound
Compound ID
CP0437159
Compound Name
(2R,3R,4S,5R)-2-[2-chloro-6-(4-chloro-2-fluoroanilino)purin-9-yl]-5-[(3,5-dimethylpyrazol-1-yl)methyl]oxolane-3,4-diol
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Structure
Formula
C21H20Cl2FN7O3
Molecular Weight
508.341
Canonical SMILES
Cc1cc(C)n(C[C@H]2O[C@H]([C@H](O)[C@@H]2O)n2cnc3c(Nc4ccc(Cl)cc4F)nc(Cl)nc23)n1
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InChI
InChI=1S/C21H20Cl2FN7O3/c1-9-5-10(2)31(29-9)7-14-16(32)17(33)20(34-14)30-8-25-15-18(27-21(23)28-19(15)30)26-13-4-3-11(22)6-12(13)24/h3-6,8,14,16-17,20,32-33H,7H2,1-2H3,(H,26,27,28)/t14-,16-,17-,20-/m1/s1
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InChIKey
BHLZQOKQEWHIPN-WVSUBDOOSA-N
Physicochemical Property
logP
3.14854
Rotatable Bonds
5
Heavy Atom Count
34
Polar Areas
123.14
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
10
Complexity
34

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 137652383
ChEMBL ID
CHEMBL4078360
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00840, Adenosine receptor A1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
EC50 = 5570 nM
   TI
   LI
   LO
   TS
2
Ki = 139 nM
   TI
   LI
   LO
   TS
Protein ID: PT00862, Adenosine receptor A2a
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
Protein ID: PT01278, Adenosine receptor A2b
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 > 60000 nM
   TI
   LI
   LO
   TS
Protein ID: PT01279, Adenosine receptor A3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 701 nM
   TI
   LI
   LO
   TS
2
Ki = 139 nM
   TI
   LI
   LO
   TS