General Information of the Compound
Compound ID
CP0434557
Compound Name
(3R)-N-[2-(4-methylphenyl)ethyl]-1-pyrimidin-2-ylpiperidine-3-carboxamide
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Structure
Formula
C19H24N4O
Molecular Weight
324.428
Canonical SMILES
Cc1ccc(CCNC(=O)[C@@H]2CCCN(C2)c2ncccn2)cc1
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InChI
InChI=1S/C19H24N4O/c1-15-5-7-16(8-6-15)9-12-20-18(24)17-4-2-13-23(14-17)19-21-10-3-11-22-19/h3,5-8,10-11,17H,2,4,9,12-14H2,1H3,(H,20,24)/t17-/m1/s1
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InChIKey
PAILKZHTLKRXQL-QGZVFWFLSA-N
Physicochemical Property
logP
2.36032
Rotatable Bonds
5
Heavy Atom Count
24
Polar Areas
58.12
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
4
Complexity
24

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 90654572
ChEMBL ID
CHEMBL3234553
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT04975, G-protein coupled bile acid receptor 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat Homo sapiens (Human)  1
1
EC50 = 2170 nM
   TI
   LI
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   TS
Protein ID: PT02509, G-protein coupled bile acid receptor 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat Homo sapiens (Human)  1
1
EC50 = 4300 nM
   TI
   LI
   LO
   TS