General Information of the Compound
Compound ID
CP0433523
Compound Name
2-[2-(5-cyano-3-hydroxy-4-methylpyridin-2-yl)-5-phenyl-1,3-thiazol-4-yl]-N-(2-pyridin-2-ylethyl)acetamide
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Structure
Formula
C25H21N5O2S
Molecular Weight
455.543
Canonical SMILES
Cc1c(O)c(ncc1C#N)-c1nc(CC(=O)NCCc2ccccn2)c(s1)-c1ccccc1
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InChI
InChI=1S/C25H21N5O2S/c1-16-18(14-26)15-29-22(23(16)32)25-30-20(24(33-25)17-7-3-2-4-8-17)13-21(31)28-12-10-19-9-5-6-11-27-19/h2-9,11,15,32H,10,12-13H2,1H3,(H,28,31)
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InChIKey
ICUKKSACAFOILF-UHFFFAOYSA-N
Physicochemical Property
logP
4.0542
Rotatable Bonds
7
Heavy Atom Count
33
Polar Areas
111.79
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
33

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 136074312
ChEMBL ID
CHEMBL3310404
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02612, Egl nine homolog 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000273 Hep 3B2.1-7 Homo sapiens (Human)  1
1
IC50 = 5700 nM
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