General Information of the Compound
Compound ID
CP0432407
Compound Name
[(19S)-10,19-diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 4-[10-(hydroxyamino)-10-oxodecanoyl]piperazine-1-carboxylate
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Structure
Formula
C37H45N5O9
Molecular Weight
703.793
Canonical SMILES
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OC(=O)N3CCN(CC3)C(=O)CCCCCCCCC(=O)NO)cc12
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InChI
InChI=1S/C37H45N5O9/c1-3-24-25-19-23(51-36(47)41-17-15-40(16-18-41)32(44)12-10-8-6-5-7-9-11-31(43)39-49)13-14-29(25)38-33-26(24)21-42-30(33)20-28-27(34(42)45)22-50-35(46)37(28,48)4-2/h13-14,19-20,48-49H,3-12,15-18,21-22H2,1-2H3,(H,39,43)/t37-/m0/s1
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InChIKey
DXLAFUMFMFMSLO-QNGWXLTQSA-N
Physicochemical Property
logP
3.9112
Rotatable Bonds
12
Heavy Atom Count
51
Polar Areas
180.6
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
11
Complexity
51

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 145983876
ChEMBL ID
CHEMBL4250057
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00991, Histone deacetylase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 30090 nM
   TI
   LI
   LO
   TS
Protein ID: PT00995, Histone deacetylase 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 25380 nM
   TI
   LI
   LO
   TS
Protein ID: PT01213, Histone deacetylase 6
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 7020 nM
   TI
   LI
   LO
   TS