General Information of the Compound
Compound ID
CP0432134
Compound Name
US10272079, Compound 61
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Structure
Formula
C78H101Cl6N9O19S3
Molecular Weight
1777.629
Canonical SMILES
CN1C[C@@H](c2cccc(c2)S(=O)(=O)NCCOCCOCCOCCNC(=O)CC(O)(CC(=O)NCCOCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)C(=O)NCCOCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)c2cc(Cl)cc(Cl)c2C1
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InChI
InChI=1S/C78H101Cl6N9O19S3/c1-91-48-66(63-40-57(79)43-72(82)69(63)51-91)54-7-4-10-60(37-54)113(98,99)88-16-22-107-28-34-110-31-25-104-19-13-85-75(94)46-78(97,77(96)87-15-21-106-27-33-112-36-30-109-24-18-90-115(102,103)62-12-6-9-56(39-62)68-50-93(3)53-71-65(68)42-59(81)45-74(71)84)47-76(95)86-14-20-105-26-32-111-35-29-108-23-17-89-114(100,101)61-11-5-8-55(38-61)67-49-92(2)52-70-64(67)41-58(80)44-73(70)83/h4-12,37-45,66-68,88-90,97H,13-36,46-53H2,1-3H3,(H,85,94)(H,86,95)(H,87,96)/t66-,67-,68-/m0/s1
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InChIKey
RHBHZMXQVQNXBK-NLXGDKCYSA-N
Physicochemical Property
logP
7.5835
Rotatable Bonds
50
Heavy Atom Count
115
Polar Areas
338.83
Hydrogen Bond Donor Count
7
Hydrogen Bond Acceptor Count
22
Complexity
115

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118933966
ChEMBL ID
CHEMBL3906665
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03762, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 15.85 nM
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Protein ID: PT04309, Sodium/hydrogen exchanger 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000422 OK Didelphis virginiana (North American opossum)  1
1
IC50 = 100 nM
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