General Information of the Compound
Compound ID
CP0431456
Compound Name
N-[2-[(2,4-dimethoxyphenyl)methyl]-1-oxoisoquinolin-7-yl]-N'-hydroxyoctanediamide
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Structure
Formula
C26H31N3O6
Molecular Weight
481.549
Canonical SMILES
COc1ccc(Cn2ccc3ccc(NC(=O)CCCCCCC(=O)NO)cc3c2=O)c(OC)c1
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InChI
InChI=1S/C26H31N3O6/c1-34-21-12-10-19(23(16-21)35-2)17-29-14-13-18-9-11-20(15-22(18)26(29)32)27-24(30)7-5-3-4-6-8-25(31)28-33/h9-16,33H,3-8,17H2,1-2H3,(H,27,30)(H,28,31)
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InChIKey
GIKBCAFOYUWQMO-UHFFFAOYSA-N
Physicochemical Property
logP
3.8515
Rotatable Bonds
12
Heavy Atom Count
35
Polar Areas
118.89
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
7
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 122185147
ChEMBL ID
CHEMBL3601775
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00991, Histone deacetylase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 98.08 nM
   TI
   LI
   LO
   TS
Protein ID: PT00995, Histone deacetylase 3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 107.7 nM
   TI
   LI
   LO
   TS
Protein ID: PT01213, Histone deacetylase 6
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000023 BTI-Tn-5B1-4 Trichoplusia ni (Cabbage looper)  1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS