General Information of the Compound
Compound ID
CP0428712
Compound Name
1-((3R,6S)-6-(3-cyanophenyl)bicyclo[4.1.0]heptan-3-yl)-3-(3,4-difluorophenyl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea
    Show/Hide
Structure
Formula
C28H32F2N4O3S
Molecular Weight
542.652
Canonical SMILES
CS(=O)(=O)N1CCC(CN([C@@H]2CC[C@@]3(CC3C2)c2cccc(c2)C#N)C(=O)Nc2ccc(F)c(F)c2)CC1
    Show/Hide
InChI
InChI=1S/C28H32F2N4O3S/c1-38(36,37)33-11-8-19(9-12-33)18-34(27(35)32-23-5-6-25(29)26(30)15-23)24-7-10-28(16-22(28)14-24)21-4-2-3-20(13-21)17-31/h2-6,13,15,19,22,24H,7-12,14,16,18H2,1H3,(H,32,35)/t22?,24-,28-/m1/s1
    Show/Hide
InChIKey
MWLQXCNQYZZYIY-FKCQOYNMSA-N
Physicochemical Property
logP
4.85238
Rotatable Bonds
6
Heavy Atom Count
38
Polar Areas
93.51
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
4
Complexity
38

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 44424231
ChEMBL ID
CHEMBL229925
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01027, Melanin-concentrating hormone receptor 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 5.4 nM
   TI
   LI
   LO
   TS