General Information of the Compound
Compound ID
CP0426771
Compound Name
(1S,2S,10R,18R)-8-benzyl-19-(cyclopropylmethyl)-2,13-dihydroxy-11-oxa-8,19-diazahexacyclo[10.9.1.01,10.02,18.04,9.016,22]docosa-4(9),12,14,16(22)-tetraen-7-one
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Structure
Formula
C30H32N2O4
Molecular Weight
484.596
Canonical SMILES
Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]45[C@@H](Oc1c24)C1=C(CCC(=O)N1Cc1ccccc1)C[C@@]35O
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InChI
InChI=1S/C30H32N2O4/c33-22-10-8-20-14-23-30(35)15-21-9-11-24(34)32(17-18-4-2-1-3-5-18)26(21)28-29(30,25(20)27(22)36-28)12-13-31(23)16-19-6-7-19/h1-5,8,10,19,23,28,33,35H,6-7,9,11-17H2/t23-,28+,29+,30-/m1/s1
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InChIKey
GTAWNDHRLYTFLJ-UJLGHMMASA-N
Physicochemical Property
logP
3.6429
Rotatable Bonds
4
Heavy Atom Count
36
Polar Areas
73.24
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
5
Complexity
36

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118705898
ChEMBL ID
CHEMBL3309515
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01200, Delta-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 0.36 nM
   TI
   LI
   LO
   TS
Protein ID: PT00983, Kappa-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 0.15 nM
   TI
   LI
   LO
   TS
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 0.18 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 1300 nM
   TI
   LI
   LO
   TS