General Information of the Compound
Compound ID
CP0423619
Compound Name
methyl N-[(1R,5R)-8-[bis(2-chlorophenyl)methyl]-3-(5-fluoropyridin-2-yl)-8-azabicyclo[3.2.1]octan-3-yl]carbamate
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Structure
Formula
C27H26Cl2FN3O2
Molecular Weight
514.428
Canonical SMILES
COC(=O)NC1(C[C@H]2CC[C@H](C1)N2C(c1ccccc1Cl)c1ccccc1Cl)c1ccc(F)cn1
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InChI
InChI=1S/C27H26Cl2FN3O2/c1-35-26(34)32-27(24-13-10-17(30)16-31-24)14-18-11-12-19(15-27)33(18)25(20-6-2-4-8-22(20)28)21-7-3-5-9-23(21)29/h2-10,13,16,18-19,25H,11-12,14-15H2,1H3,(H,32,34)/t18-,19-/m1/s1
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InChIKey
VENQODNWCYDESL-RTBURBONSA-N
Physicochemical Property
logP
6.4952
Rotatable Bonds
5
Heavy Atom Count
35
Polar Areas
54.46
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
4
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44574958
ChEMBL ID
CHEMBL511232
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 887 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 12 nM
   TI
   LI
   LO
   TS