General Information of the Compound
Compound ID
CP0417478
Compound Name
(1R,5R)-8-[bis(2-chlorophenyl)methyl]-3-piperidin-2-yl-8-azabicyclo[3.2.1]octane-3-carboxamide
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Structure
Formula
C26H31Cl2N3O
Molecular Weight
472.46
Canonical SMILES
NC(=O)C1(C[C@H]2CC[C@H](C1)N2C(c1ccccc1Cl)c1ccccc1Cl)C1CCCCN1
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InChI
InChI=1S/C26H31Cl2N3O/c27-21-9-3-1-7-19(21)24(20-8-2-4-10-22(20)28)31-17-12-13-18(31)16-26(15-17,25(29)32)23-11-5-6-14-30-23/h1-4,7-10,17-18,23-24,30H,5-6,11-16H2,(H2,29,32)/t17-,18-,23?/m1/s1
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InChIKey
LIGAXKWGEDSCQR-JGUPTHKFSA-N
Physicochemical Property
logP
5.3234
Rotatable Bonds
5
Heavy Atom Count
32
Polar Areas
58.36
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
3
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44575043
ChEMBL ID
CHEMBL512962
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 474 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 17 nM
   TI
   LI
   LO
   TS