General Information of the Compound
Compound ID
CP0416220
Compound Name
(1R,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol
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Structure
Formula
C26H21Cl2N5O2
Molecular Weight
506.393
Canonical SMILES
O[C@@H]1[C@@H]2C[C@@H]2[C@H]([C@@H]1O)n1cnc2c(NCc3cccc(Cl)c3)nc(nc12)C#Cc1cccc(Cl)c1
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InChI
InChI=1S/C26H21Cl2N5O2/c27-16-5-1-3-14(9-16)7-8-20-31-25(29-12-15-4-2-6-17(28)10-15)21-26(32-20)33(13-30-21)22-18-11-19(18)23(34)24(22)35/h1-6,9-10,13,18-19,22-24,34-35H,11-12H2,(H,29,31,32)/t18-,19+,22+,23+,24-/m0/s1
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InChIKey
JBPIBLYOBJVHKF-CQRLQNNPSA-N
Physicochemical Property
logP
4.0576
Rotatable Bonds
4
Heavy Atom Count
35
Polar Areas
96.09
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
7
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 70682887
ChEMBL ID
CHEMBL2089344
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00862, Adenosine receptor A2a
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 1800 nM
   TI
   LI
   LO
   TS
Protein ID: PT01279, Adenosine receptor A3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 210 nM
   TI
   LI
   LO
   TS