General Information of the Compound
Compound ID
CP0415027
Compound Name
4-[6-Methoxy-7-(2-piperazin-1-yl-ethoxy)-quinazolin-4-yl]-piperazine-1-carboxylic acid (4-cyano-phenyl)-amide
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Structure
Formula
C27H32N8O3
Molecular Weight
516.606
Canonical SMILES
COc1cc2c(ncnc2cc1OCCN1CCNCC1)N1CCN(CC1)C(=O)Nc1ccc(cc1)C#N
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InChI
InChI=1S/C27H32N8O3/c1-37-24-16-22-23(17-25(24)38-15-14-33-8-6-29-7-9-33)30-19-31-26(22)34-10-12-35(13-11-34)27(36)32-21-4-2-20(18-28)3-5-21/h2-5,16-17,19,29H,6-15H2,1H3,(H,32,36)
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InChIKey
AYUNZMXVGUBBHP-UHFFFAOYSA-N
Physicochemical Property
logP
2.14818
Rotatable Bonds
7
Heavy Atom Count
38
Polar Areas
118.88
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
9
Complexity
38

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 10885776
SID: 15932035
ChEMBL ID
CHEMBL338623
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00844, Platelet-derived growth factor receptor beta
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000197 MG-63 Homo sapiens (Human)  2
1
IC50 = 6500 nM
   TI
   LI
   LO
   TS
2
IC50 = 7790 nM
   TI
   LI
   LO
   TS