General Information of the Compound
Compound ID
CP0409938
Compound Name
4-fluoro-3-[[6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinazolin-4-yl]amino]-2-methylphenol
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Structure
Formula
C24H30FN5O3
Molecular Weight
455.534
Canonical SMILES
COc1cc2c(Nc3c(F)ccc(O)c3C)ncnc2cc1OCCCN1CCN(C)CC1
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InChI
InChI=1S/C24H30FN5O3/c1-16-20(31)6-5-18(25)23(16)28-24-17-13-21(32-3)22(14-19(17)26-15-27-24)33-12-4-7-30-10-8-29(2)9-11-30/h5-6,13-15,31H,4,7-12H2,1-3H3,(H,26,27,28)
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InChIKey
PZSVADNOJUBASZ-UHFFFAOYSA-N
Physicochemical Property
logP
3.55142
Rotatable Bonds
8
Heavy Atom Count
33
Polar Areas
82.98
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
8
Complexity
33

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118112080
ChEMBL ID
CHEMBL3800348
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00864, Vascular endothelial growth factor receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
IC50 > 10000 nM
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