General Information of the Compound
Compound ID
CP0402036
Compound Name
(1S,2R)-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-1-(4-fluorophenyl)-7-(4-(hydroxymethyl)phenyl)-2,3,8,8a-tetrahydroindolizin-5(1H)-one
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Structure
Formula
C31H26F7NO3
Molecular Weight
593.539
Canonical SMILES
C[C@@H](O[C@H]1CN2C(CC(=CC2=O)c2ccc(CO)cc2)[C@@H]1c1ccc(F)cc1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
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InChI
InChI=1S/C31H26F7NO3/c1-17(21-10-23(30(33,34)35)14-24(11-21)31(36,37)38)42-27-15-39-26(29(27)20-6-8-25(32)9-7-20)12-22(13-28(39)41)19-4-2-18(16-40)3-5-19/h2-11,13-14,17,26-27,29,40H,12,15-16H2,1H3/t17-,26?,27+,29+/m1/s1
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InChIKey
NJWUPRCNXYNBNF-QGYSTOEISA-N
Physicochemical Property
logP
7.2837
Rotatable Bonds
6
Heavy Atom Count
42
Polar Areas
49.77
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
3
Complexity
42

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 46884434
ChEMBL ID
CHEMBL1090288
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01410, Substance-P receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 0.39 nM
   TI
   LI
   LO
   TS
2
IC50 = 23 nM
   TI
   LI
   LO
   TS