General Information of the Compound
Compound ID
CP0393836
Compound Name
methyl 3-[(3R)-2,5-dioxo-8-[(2-phenylmethoxyacetyl)amino]-7-[2,4,5-trichloro-3-(dimethylamino)phenoxy]-3,4-dihydro-1H-1,4-benzodiazepin-3-yl]propanoate
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Structure
Formula
C30H29Cl3N4O7
Molecular Weight
663.942
Canonical SMILES
COC(=O)CC[C@H]1NC(=O)c2cc(Oc3cc(Cl)c(Cl)c(N(C)C)c3Cl)c(NC(=O)COCc3ccccc3)cc2NC1=O
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InChI
InChI=1S/C30H29Cl3N4O7/c1-37(2)28-26(32)18(31)12-23(27(28)33)44-22-11-17-20(36-30(41)19(35-29(17)40)9-10-25(39)42-3)13-21(22)34-24(38)15-43-14-16-7-5-4-6-8-16/h4-8,11-13,19H,9-10,14-15H2,1-3H3,(H,34,38)(H,35,40)(H,36,41)/t19-/m1/s1
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InChIKey
PITIBRHGTCSCNW-LJQANCHMSA-N
Physicochemical Property
logP
5.6641
Rotatable Bonds
11
Heavy Atom Count
44
Polar Areas
135.3
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
8
Complexity
44

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 137636592
ChEMBL ID
CHEMBL4061018
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03645, Nucleotide-binding oligomerization domain-containing protein 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000870 HEK-Blue Null1-v Homo sapiens (Human)  1
1
IC50 = 1330 nM
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Protein ID: PT03970, Nucleotide-binding oligomerization domain-containing protein 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000870 HEK-Blue Null1-v Homo sapiens (Human)  1
1
IC50 = 3780 nM
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