General Information of the Compound
Compound ID
CP0390803
Compound Name
(1S,2R)-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-1-(4-fluorophenyl)-2,3,8,8a-tetrahydroindolizin-5(1H)-one
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Structure
Formula
C24H20F7NO2
Molecular Weight
487.415
Canonical SMILES
C[C@@H](O[C@H]1CN2C(CC=CC2=O)[C@@H]1c1ccc(F)cc1)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
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InChI
InChI=1S/C24H20F7NO2/c1-13(15-9-16(23(26,27)28)11-17(10-15)24(29,30)31)34-20-12-32-19(3-2-4-21(32)33)22(20)14-5-7-18(25)8-6-14/h2,4-11,13,19-20,22H,3,12H2,1H3/t13-,19?,20+,22+/m1/s1
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InChIKey
MIUIONPWXDNWET-RMXHKDRNSA-N
Physicochemical Property
logP
6.264
Rotatable Bonds
4
Heavy Atom Count
34
Polar Areas
29.54
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
2
Complexity
34

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 46884430
ChEMBL ID
CHEMBL1092755
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01410, Substance-P receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 0.013 nM
   TI
   LI
   LO
   TS
2
IC50 = 0.53 nM
   TI
   LI
   LO
   TS