General Information of the Compound
Compound ID
CP0383312
Compound Name
(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol
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Structure
Formula
C26H20ClF2N5O2
Molecular Weight
507.928
Canonical SMILES
O[C@@H]1[C@@H]2C[C@@H]2[C@H]([C@@H]1O)n1cnc2c(NCc3cccc(Cl)c3)nc(nc12)C#Cc1ccc(F)c(F)c1
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InChI
InChI=1S/C26H20ClF2N5O2/c27-15-3-1-2-14(8-15)11-30-25-21-26(34(12-31-21)22-16-10-17(16)23(35)24(22)36)33-20(32-25)7-5-13-4-6-18(28)19(29)9-13/h1-4,6,8-9,12,16-17,22-24,35-36H,10-11H2,(H,30,32,33)/t16-,17+,22+,23+,24-/m0/s1
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InChIKey
XKRDCKIVPOWNFM-QSJAHPCTSA-N
Physicochemical Property
logP
3.6824
Rotatable Bonds
4
Heavy Atom Count
36
Polar Areas
96.09
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
7
Complexity
36

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 70693390
ChEMBL ID
CHEMBL2089342
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00862, Adenosine receptor A2a
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 1350 nM
   TI
   LI
   LO
   TS
Protein ID: PT01279, Adenosine receptor A3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 100 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki >= 99 nM