General Information of the Compound
Compound ID
CP0376868
Compound Name
3-[[7-[2-(1,1-dioxo-1,4-thiazinan-4-yl)ethoxy]-6-methoxyquinazolin-4-yl]amino]-4-fluoro-2-methylphenol
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Structure
Formula
C22H25FN4O5S
Molecular Weight
476.53
Canonical SMILES
COc1cc2c(Nc3c(F)ccc(O)c3C)ncnc2cc1OCCN1CCS(=O)(=O)CC1
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InChI
InChI=1S/C22H25FN4O5S/c1-14-18(28)4-3-16(23)21(14)26-22-15-11-19(31-2)20(12-17(15)24-13-25-22)32-8-5-27-6-9-33(29,30)10-7-27/h3-4,11-13,28H,5-10H2,1-2H3,(H,24,25,26)
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InChIKey
SBXFXKJOURISNO-UHFFFAOYSA-N
Physicochemical Property
logP
2.64432
Rotatable Bonds
7
Heavy Atom Count
33
Polar Areas
113.88
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
9
Complexity
33

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 127046108
ChEMBL ID
CHEMBL3797561
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00864, Vascular endothelial growth factor receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
IC50 > 10000 nM
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