General Information of the Compound
Compound ID
CP0375148
Compound Name
(R)-2-[(2S,3S)-3-{4-[2-Ethyl-5-(4-propoxy-benzyl)-2H-pyrazol-3-yl]-piperidin-1-ylmethyl}-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-3-methyl-butyric acid
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Structure
Formula
C36H49FN4O3
Molecular Weight
604.811
Canonical SMILES
CCCOc1ccc(Cc2cc(C3CCN(C[C@H]4CN(C[C@@H]4c4cccc(F)c4)[C@H](C(C)C)C(O)=O)CC3)n(CC)n2)cc1
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InChI
InChI=1S/C36H49FN4O3/c1-5-18-44-32-12-10-26(11-13-32)19-31-21-34(41(6-2)38-31)27-14-16-39(17-15-27)22-29-23-40(35(25(3)4)36(42)43)24-33(29)28-8-7-9-30(37)20-28/h7-13,20-21,25,27,29,33,35H,5-6,14-19,22-24H2,1-4H3,(H,42,43)/t29-,33+,35+/m0/s1
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InChIKey
YYKXMAVSPFGIFC-HMQVCXRFSA-N
Physicochemical Property
logP
6.4259
Rotatable Bonds
13
Heavy Atom Count
44
Polar Areas
70.83
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
6
Complexity
44

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 516191
ChEMBL ID
CHEMBL369278
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00903, C-C chemokine receptor type 5
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 0.8 nM
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