General Information of the Compound
Compound ID
CP0373376
Compound Name
(R)-2-[(2S,3S)-3-{4-[5-(3-Cyano-4-methoxy-benzyl)-2-ethyl-2H-pyrazol-3-yl]-piperidin-1-ylmethyl}-4-(3-fluoro-phenyl)-pyrrolidin-1-yl]-3-methyl-butyric acid
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Structure
Formula
C35H44FN5O3
Molecular Weight
601.767
Canonical SMILES
CCn1nc(Cc2ccc(OC)c(c2)C#N)cc1C1CCN(C[C@H]2CN(C[C@@H]2c2cccc(F)c2)[C@H](C(C)C)C(O)=O)CC1
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InChI
InChI=1S/C35H44FN5O3/c1-5-41-32(18-30(38-41)16-24-9-10-33(44-4)27(15-24)19-37)25-11-13-39(14-12-25)20-28-21-40(34(23(2)3)35(42)43)22-31(28)26-7-6-8-29(36)17-26/h6-10,15,17-18,23,25,28,31,34H,5,11-14,16,20-22H2,1-4H3,(H,42,43)/t28-,31+,34+/m0/s1
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InChIKey
RLMKPCDGHIJQNP-LKQHQURMSA-N
Physicochemical Property
logP
5.51738
Rotatable Bonds
11
Heavy Atom Count
44
Polar Areas
94.62
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
7
Complexity
44

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 516200
ChEMBL ID
CHEMBL366492
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00903, C-C chemokine receptor type 5
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 0.8 nM
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