General Information of the Compound
Compound ID
CP0372858
Compound Name
3-(cyclohexylmethyl)-8-(diphenylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
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Structure
Formula
C33H39N3O
Molecular Weight
493.695
Canonical SMILES
O=C1N(CC2CCCCC2)CN(c2ccccc2)C11CCN(CC1)C(c1ccccc1)c1ccccc1
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InChI
InChI=1S/C33H39N3O/c37-32-33(36(30-19-11-4-12-20-30)26-35(32)25-27-13-5-1-6-14-27)21-23-34(24-22-33)31(28-15-7-2-8-16-28)29-17-9-3-10-18-29/h2-4,7-12,15-20,27,31H,1,5-6,13-14,21-26H2
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InChIKey
KBHDMWWWVBHMBD-UHFFFAOYSA-N
Physicochemical Property
logP
6.4972
Rotatable Bonds
6
Heavy Atom Count
37
Polar Areas
26.79
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
3
Complexity
37

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 25190577
ChEMBL ID
CHEMBL515554
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00983, Kappa-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 2316 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 89 nM
   TI
   LI
   LO
   TS